Researcher List Hiroya Kou Hiroya Kou (廣谷 功) Please select the form format to download from below 「Education and research environment」format 「No. 4, the Ministry of Education document style ①Outline for Vitae」format 「No. 4, the Ministry of Education document style ②Education and research environment」format 「List of Teachers」format Profile Information AffiliationProfessor, Faculty of Pharmacy Department of Pharmaceutical Sciences, Musashino UniversityDegree薬学士(東北大学)薬学修士(東北大学)薬学博士(東北大学)J-GLOBAL ID201701020116661251researchmap Member IDB000270515External linkhttp://www.musashino-u.ac.jp/facilities/pharmacy/yakka.html●趣味 日曜大工,映画・海外ドラマ鑑賞,野球観戦. ●モットー やる時はやる.一心不乱. ●授業方針 基礎から応用までを丁寧に解説します. 記憶より考えて答えを出す方法を解説します. Research Interests 2 Organic Chemistry 有機化学 Research Areas 4 Life sciences / Pharmaceuticals - chemistry and drug development / Nanotechnology/Materials / Synthetic organic chemistry / Life sciences / Bioorganic chemistry / Nanotechnology/Materials / Structural/physical organic chemistry / Research History 10 Apr, 2011 - Present of Pharmaceutical Sciences, Graduate School, Musashino University Apr, 2011 - Present Faculty of Pharmacy, Department of Pharmaceutical Sciences, Musashino University Apr, 2011 - Present of Pharmaceutical Sciences, Graduate School, Musashino University Apr, 1999 - Mar, 2011 Tohoku University Graduate School of Pharmaceutical Sciences Associate Professor Feb, 1996 - Mar, 1999 Tohoku University Associate Professor More Education 3 Apr, 1985 - Mar, 1988 Graduate School, Division of Pharmaceutical Sciences, Tohoku University Apr, 1983 - Mar, 1985 Graduate School, Division of Pharmaceutical Sciences, Tohoku University Mar, 1979 - Mar, 1983 Faculty of Pharmaceutical Science, Tohoku University Awards 2 May, 1997 有機合成化学協会 研究企画賞 Dec, 1992 日本薬学会東北支部 奨励賞 Papers 102 Catalytic Direct Cyclization of Alkenyl Thioester Shiori Date, Kensei Hamasaki, Karen Sunagawa, Hiroki Koyama, Chikayoshi Sebe, Kou Hiroya, Hiroki Shigehisa ACS Catalysis, 10(3) 2039-2045, Feb 7, 2020 SIMULTANEOUS FUNCTIONALIZATION AND CYCLIZATION OF 2-ETHYNYLANILINE DERIVATIVES TO INDOLES Kou Hiroya, Shin Itoh, Kiyofumi Inamoto, Hiroki Shigehisa, Takao Sakamoto HETEROCYCLES, 95(2) 920-933, Jan, 2017 Peer-reviewed Co-Catalyzed Hydroarylation of Unactivated Olefins Hiroki Shigehisa, Takuya Ano, Hiroshi Honma, Kousuke Ebisawa, Kou Hiroya ORGANIC LETTERS, 18(15) 3622-3625, Aug, 2016 Peer-reviewed Catalytic Synthesis of Saturated Oxygen Heterocycles by Hydrofunctionalization of Unactivated Olefins: Unprotected and Protected Strategies Hiroki Shigehisa, Miki Hayashi, Haruna Ohkawa, Tsuyoshi Suzuki, Hiroki Okayasu, Mayumi Mukai, Ayaka Yamazaki, Ryohei Kawai, Harue Kikuchi, Yui Satoh, Akane Fukuyama, Kou Hiroya JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 138(33) 10597-10604, Aug, 2016 Peer-reviewed Markovnikov-Selective Addition of Fluorous Solvents to Unactivated Olefins Using a Co Catalyst Hiroki Shigehisa, Harue Kikuchi, Kou Hiroya CHEMICAL & PHARMACEUTICAL BULLETIN, 64(4) 371-374, Apr, 2016 Peer-reviewed More Misc. 1 SYNTHESIS OF 4,4-DISUBSTITUTED ISOCHROMAN-3-ONE BY A TANDEM ELECTROCYCLIC-SIGMATROPIC REACTION AND ITS APPLICATION TO THE SYNTHESIS OF NATURAL-PRODUCTS K SHISHIDO, E SHITARA, H KOMATSU, K HIROYA, K FUKUMOTO, T KAMETANI HETEROCYCLES, 24(1) 250-250, Jan, 1986 Peer-reviewed Books and Other Publications 6 薬学演習 II. 基礎科学 廣谷 功 (Role: Contributor, 第II編 化学系薬学) 東京化学同人, Oct 22, 2021 現場で役に立つ! 臨床医薬品化学 廣谷 功 (Role: Contributor, 10章 免疫・アレルギー疾患とその治療薬および抗炎症薬) 化学同人, Apr 10, 2021 化学系薬学 I. 化学物質の性質と反応 廣谷 功 (Role: Contributor, 第6章 芳香族化合物 SBO29 代表的な芳香族複素間化合物の性質を芳香属性と関連づけて説明できる.) 東京化学同人, Feb 20, 2015 新編ヘテロ環化合物 展開編 坂本 尚夫, 廣谷 功 (Role: Joint author) 講談社, Nov, 2010 (ISBN: 9784061543331) ヘテロ小員環化合物,含窒素飽和5~7員環化合物,および4級塩化合物の反応性と合成について記述した.また,芳香ヘテロ環化合物の環変換と遷移金属触媒を用いる芳香ヘテロ環への官能基導入法と閉環反応に関しても記述した. 芳香族ヘテロ環化合物の化学 -反応性と環合成- 坂本尚夫, 廣谷 功 (Role: Joint author) 講談社, Oct, 2008 (ISBN: 9784061536838) 芳香族ヘテロ環化合物の性質,反応性,官能基導入部,環合成方法などに関して記述した著書. More Presentations 55 温和な条件下でのチオエーテル含有オキサゾリン合成法の開発 長尾 芳大, 廣谷 功 第64回 日本薬学会関東支部大会, Sep, 2020 ベンジル位不斉第四級炭素構築法の開発と合成化学的応用 三嶽 香穂, 天野 智喬, 村田 いぶき, 重久 浩樹, 長尾 芳大, 廣谷 功 第64回 日本薬学会関東支部大会, Sep, 2020 アルケニルチオエステルの分子内ヒドロチオ化反応 (2):基質適用範囲の拡大 館 志織, 小山 寛貴, 瀬部 謹儀, 廣谷 功, 重久 浩樹 日本薬学会 第140年会(京都), Mar, 2020 アルケニルチオエステルの分子内ヒドロチオ化反応 (1):チオエステルの求核性 濱崎 健生, 砂川 夏蓮, 館 志織, 廣谷 功, 重久 浩樹 日本薬学会 第140年会(京都), Mar, 2020 TM-HAT/RPC 機構を基盤にした環状ウレアおよびイソウレア合成 三股 奈央, 長井 拓哉, 寺田 吉宏, 廣谷 功, 重久 浩樹 日本薬学会 第140年会(京都), Mar, 2020 More Teaching Experience 2 構造解析学 (東北大学薬学部) 有機化学 (武蔵野大学,東北大学薬学部) Professional Memberships 4 アメリカ化学会 日本化学会 日本薬学会 有機合成化学協会 Research Projects 22 Study of the Mechanism for Diastereoselective Ketal Formation Reaction and Its Application to the Synthetic Organic Chemistry. Grants-in-Aid for Scientific Research Grant-in-Aid for Scientific Research (C), Japan Society for the Promotion of Science, Apr, 2022 - Mar, 2025 Kou Hiroya Development of Chiral Ligand Containing Indazole Ring and Its Application to Dynamic Kinetic Resolution Grants-in-Aid for Scientific Research Grant-in-Aid for Scientific Research (C), Japan Society for the Promotion of Science, Apr, 2018 - Mar, 2022 Hiroya Kou Elucidation of drug interaction mechanism by metronidazole and investigation of possibility of unknown interactions. Grants-in-Aid for Scientific Research Grant-in-Aid for Young Scientists (B), Japan Society for the Promotion of Science, Apr, 2016 - Mar, 2018 KUDO Toshiyuki, ITO Kiyomi, HIROYA Kou Development and Application of Diastereoselective Ketal Formation Reaction. Apr, 2015 - Mar, 2018 Kou Hiroya Development and Application of Dynamic Kinetic Resolution Catalyzed by Chiral Pai-allyl Complex Apr, 2012 - Mar, 2015 Kou Hiroya More
Hiroya Kou (廣谷 功) Please select the form format to download from below 「Education and research environment」format 「No. 4, the Ministry of Education document style ①Outline for Vitae」format 「No. 4, the Ministry of Education document style ②Education and research environment」format 「List of Teachers」format Profile Information AffiliationProfessor, Faculty of Pharmacy Department of Pharmaceutical Sciences, Musashino UniversityDegree薬学士(東北大学)薬学修士(東北大学)薬学博士(東北大学)J-GLOBAL ID201701020116661251researchmap Member IDB000270515External linkhttp://www.musashino-u.ac.jp/facilities/pharmacy/yakka.html●趣味 日曜大工,映画・海外ドラマ鑑賞,野球観戦. ●モットー やる時はやる.一心不乱. ●授業方針 基礎から応用までを丁寧に解説します. 記憶より考えて答えを出す方法を解説します. Research Interests 2 Organic Chemistry 有機化学 Research Areas 4 Life sciences / Pharmaceuticals - chemistry and drug development / Nanotechnology/Materials / Synthetic organic chemistry / Life sciences / Bioorganic chemistry / Nanotechnology/Materials / Structural/physical organic chemistry / Research History 10 Apr, 2011 - Present of Pharmaceutical Sciences, Graduate School, Musashino University Apr, 2011 - Present Faculty of Pharmacy, Department of Pharmaceutical Sciences, Musashino University Apr, 2011 - Present of Pharmaceutical Sciences, Graduate School, Musashino University Apr, 1999 - Mar, 2011 Tohoku University Graduate School of Pharmaceutical Sciences Associate Professor Feb, 1996 - Mar, 1999 Tohoku University Associate Professor More Education 3 Apr, 1985 - Mar, 1988 Graduate School, Division of Pharmaceutical Sciences, Tohoku University Apr, 1983 - Mar, 1985 Graduate School, Division of Pharmaceutical Sciences, Tohoku University Mar, 1979 - Mar, 1983 Faculty of Pharmaceutical Science, Tohoku University Awards 2 May, 1997 有機合成化学協会 研究企画賞 Dec, 1992 日本薬学会東北支部 奨励賞 Papers 102 Catalytic Direct Cyclization of Alkenyl Thioester Shiori Date, Kensei Hamasaki, Karen Sunagawa, Hiroki Koyama, Chikayoshi Sebe, Kou Hiroya, Hiroki Shigehisa ACS Catalysis, 10(3) 2039-2045, Feb 7, 2020 SIMULTANEOUS FUNCTIONALIZATION AND CYCLIZATION OF 2-ETHYNYLANILINE DERIVATIVES TO INDOLES Kou Hiroya, Shin Itoh, Kiyofumi Inamoto, Hiroki Shigehisa, Takao Sakamoto HETEROCYCLES, 95(2) 920-933, Jan, 2017 Peer-reviewed Co-Catalyzed Hydroarylation of Unactivated Olefins Hiroki Shigehisa, Takuya Ano, Hiroshi Honma, Kousuke Ebisawa, Kou Hiroya ORGANIC LETTERS, 18(15) 3622-3625, Aug, 2016 Peer-reviewed Catalytic Synthesis of Saturated Oxygen Heterocycles by Hydrofunctionalization of Unactivated Olefins: Unprotected and Protected Strategies Hiroki Shigehisa, Miki Hayashi, Haruna Ohkawa, Tsuyoshi Suzuki, Hiroki Okayasu, Mayumi Mukai, Ayaka Yamazaki, Ryohei Kawai, Harue Kikuchi, Yui Satoh, Akane Fukuyama, Kou Hiroya JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 138(33) 10597-10604, Aug, 2016 Peer-reviewed Markovnikov-Selective Addition of Fluorous Solvents to Unactivated Olefins Using a Co Catalyst Hiroki Shigehisa, Harue Kikuchi, Kou Hiroya CHEMICAL & PHARMACEUTICAL BULLETIN, 64(4) 371-374, Apr, 2016 Peer-reviewed More Misc. 1 SYNTHESIS OF 4,4-DISUBSTITUTED ISOCHROMAN-3-ONE BY A TANDEM ELECTROCYCLIC-SIGMATROPIC REACTION AND ITS APPLICATION TO THE SYNTHESIS OF NATURAL-PRODUCTS K SHISHIDO, E SHITARA, H KOMATSU, K HIROYA, K FUKUMOTO, T KAMETANI HETEROCYCLES, 24(1) 250-250, Jan, 1986 Peer-reviewed Books and Other Publications 6 薬学演習 II. 基礎科学 廣谷 功 (Role: Contributor, 第II編 化学系薬学) 東京化学同人, Oct 22, 2021 現場で役に立つ! 臨床医薬品化学 廣谷 功 (Role: Contributor, 10章 免疫・アレルギー疾患とその治療薬および抗炎症薬) 化学同人, Apr 10, 2021 化学系薬学 I. 化学物質の性質と反応 廣谷 功 (Role: Contributor, 第6章 芳香族化合物 SBO29 代表的な芳香族複素間化合物の性質を芳香属性と関連づけて説明できる.) 東京化学同人, Feb 20, 2015 新編ヘテロ環化合物 展開編 坂本 尚夫, 廣谷 功 (Role: Joint author) 講談社, Nov, 2010 (ISBN: 9784061543331) ヘテロ小員環化合物,含窒素飽和5~7員環化合物,および4級塩化合物の反応性と合成について記述した.また,芳香ヘテロ環化合物の環変換と遷移金属触媒を用いる芳香ヘテロ環への官能基導入法と閉環反応に関しても記述した. 芳香族ヘテロ環化合物の化学 -反応性と環合成- 坂本尚夫, 廣谷 功 (Role: Joint author) 講談社, Oct, 2008 (ISBN: 9784061536838) 芳香族ヘテロ環化合物の性質,反応性,官能基導入部,環合成方法などに関して記述した著書. More Presentations 55 温和な条件下でのチオエーテル含有オキサゾリン合成法の開発 長尾 芳大, 廣谷 功 第64回 日本薬学会関東支部大会, Sep, 2020 ベンジル位不斉第四級炭素構築法の開発と合成化学的応用 三嶽 香穂, 天野 智喬, 村田 いぶき, 重久 浩樹, 長尾 芳大, 廣谷 功 第64回 日本薬学会関東支部大会, Sep, 2020 アルケニルチオエステルの分子内ヒドロチオ化反応 (2):基質適用範囲の拡大 館 志織, 小山 寛貴, 瀬部 謹儀, 廣谷 功, 重久 浩樹 日本薬学会 第140年会(京都), Mar, 2020 アルケニルチオエステルの分子内ヒドロチオ化反応 (1):チオエステルの求核性 濱崎 健生, 砂川 夏蓮, 館 志織, 廣谷 功, 重久 浩樹 日本薬学会 第140年会(京都), Mar, 2020 TM-HAT/RPC 機構を基盤にした環状ウレアおよびイソウレア合成 三股 奈央, 長井 拓哉, 寺田 吉宏, 廣谷 功, 重久 浩樹 日本薬学会 第140年会(京都), Mar, 2020 More Teaching Experience 2 構造解析学 (東北大学薬学部) 有機化学 (武蔵野大学,東北大学薬学部) Professional Memberships 4 アメリカ化学会 日本化学会 日本薬学会 有機合成化学協会 Research Projects 22 Study of the Mechanism for Diastereoselective Ketal Formation Reaction and Its Application to the Synthetic Organic Chemistry. Grants-in-Aid for Scientific Research Grant-in-Aid for Scientific Research (C), Japan Society for the Promotion of Science, Apr, 2022 - Mar, 2025 Kou Hiroya Development of Chiral Ligand Containing Indazole Ring and Its Application to Dynamic Kinetic Resolution Grants-in-Aid for Scientific Research Grant-in-Aid for Scientific Research (C), Japan Society for the Promotion of Science, Apr, 2018 - Mar, 2022 Hiroya Kou Elucidation of drug interaction mechanism by metronidazole and investigation of possibility of unknown interactions. Grants-in-Aid for Scientific Research Grant-in-Aid for Young Scientists (B), Japan Society for the Promotion of Science, Apr, 2016 - Mar, 2018 KUDO Toshiyuki, ITO Kiyomi, HIROYA Kou Development and Application of Diastereoselective Ketal Formation Reaction. Apr, 2015 - Mar, 2018 Kou Hiroya Development and Application of Dynamic Kinetic Resolution Catalyzed by Chiral Pai-allyl Complex Apr, 2012 - Mar, 2015 Kou Hiroya More